| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor M4 |
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| Ligand | BDBM82379 |
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| Substrate/Competitor | n/a |
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| Ki | 2.04±n/a nM |
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| Comments | PDSP_3897 |
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| Citation |  Lazareno, S; Buckley, NJ; Roberts, FF Characterization of muscarinic M4 binding sites in rabbit lung, chicken heart, and NG108-15 cells. Mol Pharmacol38:805-15 (1990) [PubMed] |
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| More Info.: | Get all data from this article |
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| Muscarinic acetylcholine receptor M4 |
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| Name: | Muscarinic acetylcholine receptor M4 |
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| Synonyms: | ACM4_CHICK | CHRM4 | Cholinergic, muscarinic M4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 54968.10 |
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| Organism: | Chick |
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| Description: | Cholinergic, muscarinic M4 CHRM4 Chick::P17200 |
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| Residue: | 490 |
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| Sequence: | MHNLSAQPWQAKMANLTYDNVTLSNRSEVAIQPPTNYKTVELVFIATVTGSLSLVTVVGN
ILVMLSIKVNRQLQTVNNYFLFSLACADLIIGVFSMNLYTVYIIKGYWPLGAVVCDLWLA
LDYVVSNASVMNLLIISFDRYFCVTKPLTYPARRTTKMAGLMIAAAWILSFILWAPAILF
WQFIVGKRTVHERECYIQFLSNPAVTFGTAIAAFYLPVVIMTVLYIHISLASRSRVRRHK
PESRKERKGKSLSFFKAPPVKQNNNNSPKRAVEVKEEVRNGKVDDQPSAQTEATGQQEEK
ETSNESSTVSMTQTTKDKPTTEILPAGQGQSPAHPRVNPTSKWSKIKIVTKQTGTESVTA
IEIVPAKAGASDHNSLSNSRPANVARKFASIARSQVRKKRQMAAREKKVTRTIFAILLAF
ILTWTPYNVMVLINTFCETCVPETVWSIGYWLCYVNSTINPACYALCNATFKKTFKHLLM
CQYRNIGTAR
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| BDBM82379 |
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| n/a |
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| Name | BDBM82379 |
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| Synonyms: | BTM 1042 hydrochloride | BTM1086 | CAS_87687-13-6 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H25N3OS |
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| Mol. Mass. | 367.508 |
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| SMILES | CN1CCN(C[C@@H]2[C@@H](Sc3ccccc3NC2=O)c2ccccc2)CC1 |
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| Structure | 
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