| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor |
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| Ligand | BDBM50064176 |
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| Substrate/Competitor | n/a |
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| Ki | 15.49±n/a nM |
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| Comments | PDSP_1220 |
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| Citation |  Lazareno, S; Buckley, NJ; Roberts, FF Characterization of muscarinic M4 binding sites in rabbit lung, chicken heart, and NG108-15 cells. Mol Pharmacol38:805-15 (1990) [PubMed] |
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| More Info.: | Get all data from this article |
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| Muscarinic acetylcholine receptor |
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| Name: | Muscarinic acetylcholine receptor |
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| Synonyms: | CHRM4 | Cholinergic, muscarinic M4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 53017.26 |
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| Organism: | RABBIT |
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| Description: | Cholinergic, muscarinic M4 CHRM4 RABBIT::PPPPPP |
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| Residue: | 478 |
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| Sequence: | MANFTPVNGSSSNQSVRLVTSAHNRYETVEMVFIATVTGSLSLVTVVGNVLVMLSIKVNR
QLQTVNNYFLFSLACADLIIGAFSMNLYTVYIIKGYWPLGAVVCDLWLALDYVVSNASVM
NLLIISFDRYFCVTKPLTYPARRTTKMAGLMIAAAWVLSFVLWAPAILFWQFVVGKRTVP
DNQCFIQFLSNPAVTFGTAIAAFYLPVVIMTVLYIHISLASRSRVHKHRPEGQKEKKAKT
LAFLKSPLMKQSVKKPPPGEAAREELRNGKLEEAPPPALPPPPRPMADKDTSNESSSGSA
TQNTKERPATELSTAEATTPAMSAPPLQPRTLNPASKWSKIQIVTKQTGNECVTAIEIVP
ATPAGMRPAANVARKFASIARNQVRKKRQMAARERKVTRTIFAILLAFILTWTPYNVMVL
VNTFCQSCIPDTVWSIGYWLCYVNSTINPACYALCNATFKKTFRHLLLCQYRNIGTAR
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| BDBM50064176 |
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| n/a |
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| Name | BDBM50064176 |
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| Synonyms: | CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamino)-hexyl]-octane-1,8-diamine | N1,N8-bis(6-(2-methoxybenzylamino)hexyl)octane-1,8-diamine |
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| Type | Small organic molecule |
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| Emp. Form. | C36H62N4O2 |
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| Mol. Mass. | 582.9031 |
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| SMILES | COc1ccccc1CNCCCCCCNCCCCCCCCNCCCCCCNCc1ccccc1OC |
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| Structure | 
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