| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor |
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| Ligand | BDBM82378 |
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| Substrate/Competitor | n/a |
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| Ki | 64.57±n/a nM |
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| Comments | PDSP_3905 |
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| Citation |  Lazareno, S; Buckley, NJ; Roberts, FF Characterization of muscarinic M4 binding sites in rabbit lung, chicken heart, and NG108-15 cells. Mol Pharmacol38:805-15 (1990) [PubMed] |
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| More Info.: | Get all data from this article |
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| Muscarinic acetylcholine receptor |
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| Name: | Muscarinic acetylcholine receptor |
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| Synonyms: | CHRM4 | Cholinergic, muscarinic M4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 53017.26 |
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| Organism: | RABBIT |
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| Description: | Cholinergic, muscarinic M4 CHRM4 RABBIT::PPPPPP |
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| Residue: | 478 |
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| Sequence: | MANFTPVNGSSSNQSVRLVTSAHNRYETVEMVFIATVTGSLSLVTVVGNVLVMLSIKVNR
QLQTVNNYFLFSLACADLIIGAFSMNLYTVYIIKGYWPLGAVVCDLWLALDYVVSNASVM
NLLIISFDRYFCVTKPLTYPARRTTKMAGLMIAAAWVLSFVLWAPAILFWQFVVGKRTVP
DNQCFIQFLSNPAVTFGTAIAAFYLPVVIMTVLYIHISLASRSRVHKHRPEGQKEKKAKT
LAFLKSPLMKQSVKKPPPGEAAREELRNGKLEEAPPPALPPPPRPMADKDTSNESSSGSA
TQNTKERPATELSTAEATTPAMSAPPLQPRTLNPASKWSKIQIVTKQTGNECVTAIEIVP
ATPAGMRPAANVARKFASIARNQVRKKRQMAARERKVTRTIFAILLAFILTWTPYNVMVL
VNTFCQSCIPDTVWSIGYWLCYVNSTINPACYALCNATFKKTFRHLLLCQYRNIGTAR
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| BDBM82378 |
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| n/a |
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| Name | BDBM82378 |
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| Synonyms: | CAS_82-98-4 | NSC_4839 | Piperidolate |
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| Type | Small organic molecule |
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| Emp. Form. | C21H25NO2 |
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| Mol. Mass. | 323.4287 |
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| SMILES | CCN1CCCC(C1)OC(=O)C(c1ccccc1)c1ccccc1 |
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| Structure | 
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