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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Mu-type opioid receptor | ||
| Ligand | BDBM82425 | ||
| Substrate/Competitor | n/a | ||
| Ki | 0.27±n/a nM | ||
| Comments | PDSP_806 | ||
| Citation |  Raynor, K; Kong, H; Mestek, A; Bye, LS; Tian, M; Liu, J; Yu, L; Reisine, T Characterization of the cloned human mu opioid receptor. J Pharmacol Exp Ther272:423-8 (1995) [PubMed] | ||
| More Info.: | Get all data from this article | ||
| Mu-type opioid receptor | |||
| Name: | Mu-type opioid receptor | ||
| Synonyms: | MOR-1 | MUOR1 | Mu-type opioid receptor (MOR) | OPIATE Mu | OPRM_RAT | Opiate non-selective | Opioid receptor B | Oprm1 | Ror-b | ||
| Type: | G Protein-Coupled Receptor (GPCR) | ||
| Mol. Mass.: | 44503.11 | ||
| Organism: | Rattus norvegicus (rat) | ||
| Description: | Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the mu opioid receptor. | ||
| Residue: | 398 | ||
| Sequence: |
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| BDBM82425 | |||
| n/a | |||
| Name | BDBM82425 | ||
| Synonyms: | CAS_61677 | ETORPHINE - HCI | NSC_61677 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C25H33NO4 | ||
| Mol. Mass. | 411.5338 | ||
| SMILES | CCCC(C)(O)C1CC23C=CC1(OC)C1Oc4c5c(CC2N(C)CCC315)ccc4O |c:9,TLB:16:17:8:24.23.21,7:8:24.23.21:19.18.17,9:8:24.23.21:19.18.17,THB:22:21:8:19.18.17,(7.51,1.44,;6.12,.92,;4.97,1.86,;3.58,1.33,;3.06,2.72,;4.11,-.06,;2.19,.81,;1.92,-.83,;.53,-1.78,;.54,-.47,;1.16,.67,;.87,1.89,;.87,3.38,;-.41,4.13,;-.43,.85,;-1.52,1.9,;-2.75,1.03,;-2.22,-.44,;-3.43,-1.4,;-2.64,-2.71,;-1.09,-2.63,;-1.24,-4.18,;-2.27,-5.25,;.23,-3.98,;-.13,-2.47,;-.69,-.85,;-4.92,-.98,;-5.27,.51,;-4.18,1.56,;-4.48,3.02,)| | ||
| Structure | 
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