| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 1 |
|---|
| Ligand | BDBM82454 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 1000±n/a nM |
|---|
| Comments | PDSP_1037 |
|---|
| Citation |  Hoyer, D; Lübbert, H; Bruns, C Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch Pharmacol350:441-53 (1994) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Somatostatin receptor type 1 |
|---|
| Name: | Somatostatin receptor type 1 |
|---|
| Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 42692.81 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P30872 |
|---|
| Residue: | 391 |
|---|
| Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
|
|
|
|---|
| BDBM82454 |
|---|
| n/a |
|---|
| Name | BDBM82454 |
|---|
| Synonyms: | L-363,572 | N-Methylcyclo(D-Ala-D-Phe-D-Trp-L-Lys-D-Thr-N-methyl-D-Phe-) |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C44H56N8O7 |
|---|
| Mol. Mass. | 808.9648 |
|---|
| SMILES | C[C@H](O)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](C)N(C)C(=O)[C@@H](Cc2ccccc2)N(C)C1=O |
|---|
| Structure | 
|
|---|
Search and Browse
