| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 5 |
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| Ligand | BDBM82470 |
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| Substrate/Competitor | n/a |
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| Ki | 0.10±n/a nM |
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| Comments | PDSP_373 |
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| Citation |  Hoyer, D; Lübbert, H; Bruns, C Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch Pharmacol350:441-53 (1994) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Somatostatin receptor type 5 |
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| Name: | Somatostatin receptor type 5 |
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| Synonyms: | SOMATOSTATIN SST5 | SSR5_RAT | Somatostatin receptor | Somatostatin receptor type 5 | Sstr5 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 39986.50 |
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| Organism: | RAT |
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| Description: | SOMATOSTATIN SST5 SSTR5 RAT::P30938 |
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| Residue: | 363 |
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| Sequence: | MEPLSLASTPSWNASAASSGNHNWSLVGSASPMGARAVLVPVLYLLVCTVGLSGNTLVIY
VVLRHAKMKTVTNVYILNLAVADVLFMLGLPFLATQNAVVSYWPFGSFLCRLVMTLDGIN
QFTSIFCLMVMSVDRYLAVVHPLRSARWRRPRVAKMASAAVWVFSLLMSLPLLVFADVQE
GWGTCNLSWPEPVGLWGAAFITYTSVLGFFGPLLVICLCYLLIVVKVKAAGMRVGSSRRR
RSEPKVTRMVVVVVLVFVGCWLPFFIVNIVNLAFTLPEEPTSAGLYFFVVVLSYANSCAN
PLLYGFLSDNFRQSFRKVLCLRRGYGMEDADAIEPRPDKSGRPQATLPTRSCEANGLMQT
SRI
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| BDBM82470 |
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| n/a |
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| Name | BDBM82470 |
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| Synonyms: | 3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Val-L-Cys(1)-L-Thr-NH2 | BIM 23014 | BIM-23014 | LANREOTIDE |
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| Type | Small organic molecule |
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| Emp. Form. | C54H69N11O10S2 |
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| Mol. Mass. | 1096.323 |
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| SMILES | CC(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N[C@@H]([C@@H](C)O)C(N)=O)NC(=O)[C@H](N)Cc1ccc2ccccc2c1 |
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| Structure | 
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