| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 5 |
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| Ligand | BDBM82464 |
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| Substrate/Competitor | n/a |
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| Ki | 1.58±n/a nM |
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| Comments | PDSP_1591 |
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| Citation |  Hoyer, D; Lübbert, H; Bruns, C Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch Pharmacol350:441-53 (1994) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Somatostatin receptor type 5 |
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| Name: | Somatostatin receptor type 5 |
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| Synonyms: | SOMATOSTATIN SST5 | SSR5_RAT | Somatostatin receptor | Somatostatin receptor type 5 | Sstr5 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 39986.50 |
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| Organism: | RAT |
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| Description: | SOMATOSTATIN SST5 SSTR5 RAT::P30938 |
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| Residue: | 363 |
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| Sequence: | MEPLSLASTPSWNASAASSGNHNWSLVGSASPMGARAVLVPVLYLLVCTVGLSGNTLVIY
VVLRHAKMKTVTNVYILNLAVADVLFMLGLPFLATQNAVVSYWPFGSFLCRLVMTLDGIN
QFTSIFCLMVMSVDRYLAVVHPLRSARWRRPRVAKMASAAVWVFSLLMSLPLLVFADVQE
GWGTCNLSWPEPVGLWGAAFITYTSVLGFFGPLLVICLCYLLIVVKVKAAGMRVGSSRRR
RSEPKVTRMVVVVVLVFVGCWLPFFIVNIVNLAFTLPEEPTSAGLYFFVVVLSYANSCAN
PLLYGFLSDNFRQSFRKVLCLRRGYGMEDADAIEPRPDKSGRPQATLPTRSCEANGLMQT
SRI
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| BDBM82464 |
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| n/a |
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| Name | BDBM82464 |
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| Synonyms: | CAS_71306 | NSC_71306 | RC 160 | Vapreotide |
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| Type | Small organic molecule |
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| Emp. Form. | C57H70N12O9S2 |
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| Mol. Mass. | 1131.371 |
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| SMILES | CC(C)C1NC(=O)C(CCCCN)NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C(Cc2ccc(O)cc2)NC(=O)C(CSSCC(NC1=O)C(=O)NC(Cc1c[nH]c2ccccc12)C(N)=O)NC(=O)C(N)Cc1ccccc1 |
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| Structure | 
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