| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Beta-1 adrenergic receptor |
|---|
| Ligand | BDBM25770 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | >10000±n/a nM |
|---|
| Comments | PDSP_1799 |
|---|
| Citation |  Fraundorfer, PF; Fertel, RH; Miller, DD; Feller, DR Biochemical and pharmacological characterization of high-affinity trimetoquinol analogs on guinea pig and human beta adrenergic receptor subtypes: evidence for partial agonism. J Pharmacol Exp Ther270:665-74 (1994) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Beta-1 adrenergic receptor |
|---|
| Name: | Beta-1 adrenergic receptor |
|---|
| Synonyms: | ADRB1 | Adrenergic receptor | adrenergic Beta1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 50540.48 |
|---|
| Organism: | GUINEA PIG |
|---|
| Description: | adrenergic Beta1 ADRB1 GUINEA PIG::B0FL73 |
|---|
| Residue: | 467 |
|---|
| Sequence: | MGAGVLALGASEPCNLSSTAPLPDGAATAARLLVPASPPASLLPPTSEGSEPLSPQWTAG
MGLLMVLIVLLIVAGNVLVIVAIAKTPRLQTLTNLFIMSLASADLVMGLLVVPFGATIVV
WGRWEYGSFFCELWTSVDVLCVTASIETLCVIALDRYLAITSPFRYQSLLTRARARVLVC
TVWAISALVSFLPILMHWWRAEGDEARRCYNDPKCCDFVTNRAYAIASSVVSFYVPLCIM
AFVYLRVFREAQKQVKKIDSCERRFLGGPGRPPSPVPSPTPGSPRAATDPLANGRTSKRR
PSRLVALREQKALKTLGIIMGVFTLCWLPFFLANVVKAFHRDLVPDRLFVFFNWLGYANS
AFNPIIYCRSPDFRKAFQRLLCCARRAARRRHTAHGGRPRASGCLARSGPPPSPGAASDE
DEDAVGAAPPARLLEPWAGCNGGAATADSDWSLDEPGRAGFASESKV
|
|
|
|---|
| BDBM25770 |
|---|
| n/a |
|---|
| Name | BDBM25770 |
|---|
| Synonyms: | 5-[2-(tert-butylamino)-1-hydroxyethyl]benzene-1,3-diol | 5-[2-(tert-butylamino)-1-hydroxyethyl]benzene-1,3-diol, 5 | Brethaire | Brethine | Bricanyl | Terbutaline | Terbutaline,(+/-) |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C12H19NO3 |
|---|
| Mol. Mass. | 225.2842 |
|---|
| SMILES | CC(C)(C)NCC(O)c1cc(O)cc(O)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
