| Reaction Details |
|---|
 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 1B |
|---|
| Ligand | BDBM81497 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 147.91±n/a nM |
|---|
| Comments | PDSP_491 |
|---|
| Citation |  Boess, FG; Martin, IL Molecular biology of 5-HT receptors. Neuropharmacology33:275-317 (1994) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| 5-hydroxytryptamine receptor 1B |
|---|
| Name: | 5-hydroxytryptamine receptor 1B |
|---|
| Synonyms: | 5-HT-1B | 5-HT1B | 5-hydroxytryptamine receptor 1B (5HT1B) | 5HT1B_RAT | 5ht1b | Htr1b | Serotonin 1 (5-HT1) receptor | Serotonin 1B/1D receptor | Serotonin receptor 1B |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 43173.33 |
|---|
| Organism: | Rattus norvegicus (Rat) |
|---|
| Description: | P28564 |
|---|
| Residue: | 386 |
|---|
| Sequence: | MEEQGIQCAPPPPATSQTGVPLANLSHNCSADDYIYQDSIALPWKVLLVALLALITLATT
LSNAFVIATVYRTRKLHTPANYLIASLAVTDLLVSILVMPISTMYTVTGRWTLGQVVCDF
WLSSDITCCTASIMHLCVIALDRYWAITDAVDYSAKRTPKRAAIMIVLVWVFSISISLPP
FFWRQAKAEEEVLDCFVNTDHVLYTVYSTVGAFYLPTLLLIALYGRIYVEARSRILKQTP
NKTGKRLTRAQLITDSPGSTSSVTSINSRVPEVPSESGSPVYVNQVKVRVSDALLEKKKL
MAARERKATKTLGIILGAFIVCWLPFFIISLVMPICKDACWFHMAIFDFFNWLGYLNSLI
NPIIYTMSNEDFKQAFHKLIRFKCTG
|
|
|
|---|
| BDBM81497 |
|---|
| n/a |
|---|
| Name | BDBM81497 |
|---|
| Synonyms: | 4-(4-Methyl-piperazin-1-yl)-7-trifluoromethyl-pyrrolo[1,2-a]quinoxaline | CAS_109028-10-6 | CGS 12066B | CHEMBL27403 | NSC_123945 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H17F3N4 |
|---|
| Mol. Mass. | 334.3389 |
|---|
| SMILES | CN1CCN(CC1)c1nc2cc(ccc2n2cccc12)C(F)(F)F |
|---|
| Structure | 
|
|---|
Search and Browse
