| Reaction Details |
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 | Report a problem with these data |
| Target | Transmembrane and immunoglobulin domain-containing 3 |
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| Ligand | BDBM82528 |
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| Substrate/Competitor | n/a |
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| Ki | 6.8±n/a nM |
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| Comments | PDSP_2589 |
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| Citation |  van Galen, PJ; van Bergen, AH; Gallo-Rodriguez, C; Melman, N; Olah, ME; IJzerman, AP; Stiles, GL; Jacobson, KA A binding site model and structure-activity relationships for the rat A3 adenosine receptor. Mol Pharmacol45:1101-11 (1994) [PubMed] |
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| More Info.: | Get all data from this article |
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| Transmembrane and immunoglobulin domain-containing 3 |
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| Name: | Transmembrane and immunoglobulin domain-containing 3 |
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| Synonyms: | ADENOSINE A3 | ADORA3 | Adora3 protein |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 25707.75 |
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| Organism: | RAT |
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| Description: | Q4V8H0 |
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| Residue: | 232 |
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| Sequence: | MEPLLLLSLALFSDAMVMDEKVKSGVELDTASAICNYDAHYKDHTKYWCRGYFRDSCNII
AFTPNSSNRVALKDTGDQLIITVSCLVKEDTGWYWCGIQRDFARDDMDFTKLIVTDNRED
RANGLSPGTSGNRTRSCKTSKAVQKAEGSRMSILIVCVLISGLGIIFLISHMSRGRRSQR
NRGVTGKSINRNPQASQAPSMVSIPLTVLPKVPRQNGQQKALQWTGNATKTG
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| BDBM82528 |
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| n/a |
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| Name | BDBM82528 |
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| Synonyms: | N6-BenzylNECA |
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| Type | Small organic molecule |
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| Emp. Form. | C20H24N6O5 |
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| Mol. Mass. | 428.4418 |
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| SMILES | CCNC(=O)OC[C@H]1OC([C@H](O)[C@@H]1O)n1cnc2c(NCc3ccccc3)ncnc12 |
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| Structure | 
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