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TargetCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
LigandBDBM50431
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay
IC50 5838±363 nM
Citation PubChem, PC Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,  Assay Method
 
Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
Name:Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
Synonyms:CTDS1_HUMAN | CTDSP1 | NIF3 | NLIIF | SCP1 | carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1
Type:Enzyme Catalytic Domain
Mol. Mass.:29199.89
Organism:Homo sapiens (Human)
Description:gi_10864009
Residue:261
Sequence:
MDSSAVITQISKEEARGPLRGKGDQKSAASQKPRSRGILHSLFCCVCRDDGEALPAHSGA
PLLVEENGAIPKQTPVQYLLPEAKAQDSDKICVVIDLDETLVHSSFKPVNNADFIIPVEI
DGVVHQVYVLKRPHVDEFLQRMGELFECVLFTASLAKYADPVADLLDKWGAFRARLFRES
CVFHRGNYVKDLSRLGRDLRRVLILDNSPASYVFHPDNAVPVASWFDNMSDTELHDLLPF
FEQLSRVDDVYSVLRQPRPGS
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BDBM50431
n/a
NameBDBM50431
Synonyms:(5Z)-2-azanylidene-3-(4-fluorophenyl)-5-[(4-hydroxyphenyl)methylidene]-1,3-thiazolidin-4-one | (5Z)-3-(4-fluorophenyl)-5-(4-hydroxybenzylidene)-2-imino-thiazolidin-4-one | (5Z)-3-(4-fluorophenyl)-5-[(4-hydroxyphenyl)methylidene]-2-imino-1,3-thiazolidin-4-one | (5Z)-3-(4-fluorophenyl)-5-[(4-hydroxyphenyl)methylidene]-2-imino-4-thiazolidinone | 3-(4-fluorophenyl)-5-(4-hydroxybenzylidene)-2-imino-1,3-thiazolidin-4-one | MLS000676410 | SMR000298434 | cid_1258959
TypeSmall organic molecule
Emp. Form.C16H11FN2O2S
Mol. Mass.314.334
SMILESOc1ccc(\C=C2/SC(=N)N(C2=O)c2ccc(F)cc2)cc1
Structure
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