Ki Summary

Reaction Details

Report a problem with these data

Target

Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1

Ligand

BDBM53091

Substrate/Competitor

n/a

Meas. Tech.

Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay

IC50

36102±3185 nM

Citation

PubChem, PC Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay PubChem Bioassay(2011)[AID]

More Info.:

Get all data from this article, Assay Method

Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1

Name:

Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

29199.89

Organism:

Homo sapiens (Human)

Description:

gi_10864009

Residue:

261

Sequence:

MDSSAVITQISKEEARGPLRGKGDQKSAASQKPRSRGILHSLFCCVCRDDGEALPAHSGA
PLLVEENGAIPKQTPVQYLLPEAKAQDSDKICVVIDLDETLVHSSFKPVNNADFIIPVEI
DGVVHQVYVLKRPHVDEFLQRMGELFECVLFTASLAKYADPVADLLDKWGAFRARLFRES
CVFHRGNYVKDLSRLGRDLRRVLILDNSPASYVFHPDNAVPVASWFDNMSDTELHDLLPF
FEQLSRVDDVYSVLRQPRPGS

BDBM53091

n/a

Name

BDBM53091

Synonyms:

(2E)-5-nitro-6-oxidanyl-2-[(2Z)-2-(3-oxidanyl-4-oxidanylidene-cyclohexa-2,5-dien-1-ylidene)ethylidene]-1H-pyrimidin-4-one | (2E)-6-hydroxy-2-[(2Z)-2-(3-hydroxy-4-keto-cyclohexa-2,5-dien-1-ylidene)ethylidene]-5-nitro-1H-pyrimidin-4-one | (2E)-6-hydroxy-2-[(2Z)-2-(3-hydroxy-4-oxo-1-cyclohexa-2,5-dienylidene)ethylidene]-5-nitro-1H-pyrimidin-4-one | (2E)-6-hydroxy-2-[(2Z)-2-(3-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)ethylidene]-5-nitro-1H-pyrimidin-4-one | 2-[(Z)-2-(3,4-Dihydroxy-phenyl)-vinyl]-6-hydroxy-5-nitro-3H-pyrimidin-4-one | MLS001201374 | SMR000524347 | cid_25043520

Type

Small organic molecule

Emp. Form.

C12H9N3O6

Mol. Mass.

291.2164

SMILES

Oc1[nH+]c(\C=C\[c-]2ccc(=O)c(O)c2)[nH]c(=O)c1[N+]([O-])=O

Structure