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TargetCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
LigandBDBM64129
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay
IC50 21092±2327 nM
Citation PubChem, PC Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,  Assay Method
 
Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
Name:Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
Synonyms:CTDS1_HUMAN | CTDSP1 | NIF3 | NLIIF | SCP1 | carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1
Type:Enzyme Catalytic Domain
Mol. Mass.:29199.89
Organism:Homo sapiens (Human)
Description:gi_10864009
Residue:261
Sequence:
MDSSAVITQISKEEARGPLRGKGDQKSAASQKPRSRGILHSLFCCVCRDDGEALPAHSGA
PLLVEENGAIPKQTPVQYLLPEAKAQDSDKICVVIDLDETLVHSSFKPVNNADFIIPVEI
DGVVHQVYVLKRPHVDEFLQRMGELFECVLFTASLAKYADPVADLLDKWGAFRARLFRES
CVFHRGNYVKDLSRLGRDLRRVLILDNSPASYVFHPDNAVPVASWFDNMSDTELHDLLPF
FEQLSRVDDVYSVLRQPRPGS
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  Blast E-value cutoff:
BDBM64129
n/a
NameBDBM64129
Synonyms:MLS001202278 | N-(2-ethylphenyl)-3-(4-methoxyphenyl)sulfonyl-propanamide | N-(2-ethylphenyl)-3-(4-methoxyphenyl)sulfonyl-propionamide | N-(2-ethylphenyl)-3-(4-methoxyphenyl)sulfonylpropanamide | N-(2-ethylphenyl)-3-[(4-methoxyphenyl)sulfonyl]propanamide | SMR000564981 | cid_5072004
TypeSmall organic molecule
Emp. Form.C18H21NO4S
Mol. Mass.347.429
SMILESCCc1ccccc1NC(=O)CCS(=O)(=O)c1ccc(OC)cc1
Structure
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