| Reaction Details |
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 | Report a problem with these data |
| Target | C-C chemokine receptor type 6 |
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| Ligand | BDBM80006 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | SAR analysis of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay |
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| IC50 | 9410±n/a nM |
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| Citation |  PubChem, PC SAR analysis of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| C-C chemokine receptor type 6 |
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| Name: | C-C chemokine receptor type 6 |
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| Synonyms: | C-C chemokine receptor type 6 | C-C chemokine receptor type 6 (CCR6) | CCR6 | CCR6_HUMAN | CKRL3 | CMKBR6 | GPR29 | STRL22 |
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| Type: | Enzyme |
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| Mol. Mass.: | 42510.84 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P51684 |
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| Residue: | 374 |
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| Sequence: | MSGESMNFSDVFDSSEDYFVSVNTSYYSVDSEMLLCSLQEVRQFSRLFVPIAYSLICVFG
LLGNILVVITFAFYKKARSMTDVYLLNMAIADILFVLTLPFWAVSHATGAWVFSNATCKL
LKGIYAINFNCGMLLLTCISMDRYIAIVQATKSFRLRSRTLPRSKIICLVVWGLSVIISS
STFVFNQKYNTQGSDVCEPKYQTVSEPIRWKLLMLGLELLFGFFIPLMFMIFCYTFIVKT
LVQAQNSKRHKAIRVIIAVVLVFLACQIPHNMVLLVTAANLGKMNRSCQSEKLIGYTKTV
TEVLAFLHCCLNPVLYAFIGQKFRNYFLKILKDLWCVRRKYKSSGFSCAGRYSENISRQT
SETADNDNASSFTM
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| BDBM80006 |
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| n/a |
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| Name | BDBM80006 |
|---|
| Synonyms: | 2,5-diphenyl-N'-(phenylcarbonyl)pyrazole-3-carbohydrazide | MLS000388665 | N'-benzoyl-2,5-diphenyl-3-pyrazolecarbohydrazide | N'-benzoyl-2,5-diphenyl-pyrazole-3-carbohydrazide | N'-benzoyl-2,5-diphenylpyrazole-3-carbohydrazide | SMR000254838 | cid_4883406 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H18N4O2 |
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| Mol. Mass. | 382.4146 |
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| SMILES | O=C(NNC(=O)c1ccccc1)c1cc(nn1-c1ccccc1)-c1ccccc1 |
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| Structure | 
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|---|
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