Reaction Details | |||
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Target | Phospholipase A2 | ||
Ligand | BDBM34671 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay | ||
IC50 | >80000±n/a nM | ||
Citation | PubChem, PC Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay PubChem Bioassay(2011)[AID] | ||
More Info.: | Get all data from this article, Assay Method | ||
Phospholipase A2 | |||
Name: | Phospholipase A2 | ||
Synonyms: | Group IB phospholipase A2 | PA21B_HUMAN | PLA2 | PLA2A | PLA2G1B | PPLA2 | Phosphatidylcholine 2-acylhydrolase 1B | Phospholipase A2 (PLA2) | Phospholipase A2 group 1B | phospholipase A2 precursor | ||
Type: | Protein | ||
Mol. Mass.: | 16364.13 | ||
Organism: | Homo sapiens (Human) | ||
Description: | P04054 | ||
Residue: | 148 | ||
Sequence: |
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BDBM34671 | |||
n/a | |||
Name | BDBM34671 | ||
Synonyms: | 1,3,6-Trimethyl-1H-pyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-quinone | MLS000528498 | SMR000121073 | US9073941, 611 | cid_460747 | ||
Type | Small organic molecule | ||
Emp. Form. | C8H9N5O2 | ||
Mol. Mass. | 207.1894 | ||
SMILES | Cc1nn(C)c2nc(=O)n(C)c(=O)c2n1 | ||
Structure |