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TargetPhospholipase A2
LigandBDBM34671
Substrate/Competitorn/a
Meas. Tech.Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay
IC50>80000±n/a nM
Citation PubChem, PC Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,  Assay Method
 
Phospholipase A2
Name:Phospholipase A2
Synonyms:Group IB phospholipase A2 | PA21B_HUMAN | PLA2 | PLA2A | PLA2G1B | PPLA2 | Phosphatidylcholine 2-acylhydrolase 1B | Phospholipase A2 (PLA2) | Phospholipase A2 group 1B | phospholipase A2 precursor
Type:Protein
Mol. Mass.:16364.13
Organism:Homo sapiens (Human)
Description:P04054
Residue:148
Sequence:
MKLLVLAVLLTVAAADSGISPRAVWQFRKMIKCVIPGSDPFLEYNNYGCYCGLGGSGTPV
DELDKCCQTHDNCYDQAKKLDSCKFLLDNPYTHTYSYSCSGSAITCSSKNKECEAFICNC
DRNAAICFSKAPYNKAHKNLDTKKYCQS
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BDBM34671
n/a
NameBDBM34671
Synonyms:1,3,6-Trimethyl-1H-pyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-quinone | MLS000528498 | SMR000121073 | US9073941, 611 | cid_460747
TypeSmall organic molecule
Emp. Form.C8H9N5O2
Mol. Mass.207.1894
SMILESCc1nn(C)c2nc(=O)n(C)c(=O)c2n1
Structure
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