| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Phospholipase A2 |
|---|
| Ligand | BDBM31751 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay |
|---|
| IC50 | 7530±n/a nM |
|---|
| Citation |  PubChem, PC Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay PubChem Bioassay(2011)[AID] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Phospholipase A2 |
|---|
| Name: | Phospholipase A2 |
|---|
| Synonyms: | Group IB phospholipase A2 | PA21B_HUMAN | PLA2 | PLA2A | PLA2G1B | PPLA2 | Phosphatidylcholine 2-acylhydrolase 1B | Phospholipase A2 (PLA2) | Phospholipase A2 group 1B | phospholipase A2 precursor |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 16364.13 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P04054 |
|---|
| Residue: | 148 |
|---|
| Sequence: | MKLLVLAVLLTVAAADSGISPRAVWQFRKMIKCVIPGSDPFLEYNNYGCYCGLGGSGTPV
DELDKCCQTHDNCYDQAKKLDSCKFLLDNPYTHTYSYSCSGSAITCSSKNKECEAFICNC
DRNAAICFSKAPYNKAHKNLDTKKYCQS
|
|
|
|---|
| BDBM31751 |
|---|
| n/a |
|---|
| Name | BDBM31751 |
|---|
| Synonyms: | 3-[(2-chlorobenzyl)thio]-5,6-bis(2-furyl)-1,2,4-triazine | 3-[(2-chlorophenyl)methylsulfanyl]-5,6-bis(furan-2-yl)-1,2,4-triazine | 3-[(2-chlorophenyl)methylthio]-5,6-bis(2-furanyl)-1,2,4-triazine | MLS-0002046.0001 | cid_6400942 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H12ClN3O2S |
|---|
| Mol. Mass. | 369.825 |
|---|
| SMILES | Clc1ccccc1CSc1nnc(-c2ccco2)c(n1)-c1ccco1 |
|---|
| Structure | 
|
|---|
Search and Browse
