| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM83443 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Counterscreen for agonists of heterodimerization of the mu 1 (OPRM1) and delta 1 (OPRD1) opioid receptors: Luminescence-based cell-based high throughput dose response assay |
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| EC50 | >92455±n/a nM |
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| Citation |  PubChem, PC Counterscreen for agonists of heterodimerization of the mu 1 (OPRM1) and delta 1 (OPRD1) opioid receptors: Luminescence-based cell-based high throughput dose response assay to identify agonists of OPRD1 homodimerization PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | D-OR-1 | DOR-1 | Delta opioid receptor | Delta-type opioid receptor (Delta) | OPIATE Delta | OPRD | OPRD1 | OPRD_HUMAN | OPRK1 | opioid receptor, delta 1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 40382.98 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the delta opioid receptor. |
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| Residue: | 372 |
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| Sequence: | MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTAC
TPSDGPGGGAAA
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| BDBM83443 |
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| n/a |
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| Name | BDBM83443 |
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| Synonyms: | MLS002425557 | N-[2-keto-3-methyl-1-(3-phenylpropyl)pyrrolidin-3-yl]-3,3,3-triphenyl-propionamide | N-[3-methyl-2-oxidanylidene-1-(3-phenylpropyl)pyrrolidin-3-yl]-3,3,3-triphenyl-propanamide | N-[3-methyl-2-oxo-1-(3-phenylpropyl)-3-pyrrolidinyl]-3,3,3-triphenylpropanamide | N-[3-methyl-2-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-3,3,3-triphenylpropanamide | SMR001371501 | cid_44142946 |
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| Type | Small organic molecule |
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| Emp. Form. | C35H36N2O2 |
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| Mol. Mass. | 516.6725 |
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| SMILES | CC1(CCN(CCCc2ccccc2)C1=O)NC(=O)CC(c1ccccc1)(c1ccccc1)c1ccccc1 |
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| Structure | 
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