| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 3 |
|---|
| Ligand | BDBM82463 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 30±n/a nM |
|---|
| Comments | PDSP_1033 |
|---|
| Citation |  Raynor, K; Murphy, WA; Coy, DH; Taylor, JE; Moreau, JP; Yasuda, K; Bell, GI; Reisine, T Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding of linear peptides. Mol Pharmacol43:838-44 (1993) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Somatostatin receptor type 3 |
|---|
| Name: | Somatostatin receptor type 3 |
|---|
| Synonyms: | SOMATOSTATIN SST3 | SS3R | SSR-28 | SSR3_MOUSE | Smstr3 | Somatostatin receptor | Somatostatin receptor 3 | Somatostatin receptor type 3 | Sstr3 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 47225.49 |
|---|
| Organism: | MOUSE |
|---|
| Description: | SOMATOSTATIN SST3 SSTR3 MOUSE::P30935 |
|---|
| Residue: | 428 |
|---|
| Sequence: | MATVTYPSSEPTTLDPGNASSTWPLDTTLGNTSAGASLTGLAVSGILISLVYLVVCVVGL
LGNSLVIYVVLRHTSSPSVTSVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLV
MAVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVV
VFSGVPRGMSTCHMQWPEPAAAWRTAFIIYTAALGFFGPLLVICLCYLLIVVKVRSTTRR
VRAPSCQWVQAPACQRRRRSERRVTRMVVAVVALFVLCWMPFYLLNIVNVVCPLPEEPAF
FGLYFLVVALPYANSCANPILYGFLSYRFKQGFRRILLRPSRRIRSQEPGSGPPEKTEEE
EDEEEEERREEEERRMQRGQEMNGRLSQIAQAGTSGQQPRPCTGTAKEQQLLPQEATAGD
KASTLSHL
|
|
|
|---|
| BDBM82463 |
|---|
| n/a |
|---|
| Name | BDBM82463 |
|---|
| Synonyms: | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-amino*heptanoyl-L-Phe-)] | L-362,855 | L-362855 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C57H70N10O8 |
|---|
| Mol. Mass. | 1023.2279 |
|---|
| SMILES | C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)CCCCCCNC(=O)[C@H](Cc2ccccc2)NC1=O |
|---|
| Structure | 
|
|---|
Search and Browse
