| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 4 |
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| Ligand | BDBM50065453 |
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| Substrate/Competitor | n/a |
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| Ki | 3.2±n/a nM |
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| Comments | PDSP_1035 |
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| Citation |  Raynor, K; O'Carroll, AM; Kong, H; Yasuda, K; Mahan, LC; Bell, GI; Reisine, T Characterization of cloned somatostatin receptors SSTR4 and SSTR5. Mol Pharmacol44:385-92 (1993) [PubMed] |
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| More Info.: | Get all data from this article |
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| Somatostatin receptor type 4 |
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| Name: | Somatostatin receptor type 4 |
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| Synonyms: | SOMATOSTATIN SST4 | SSR4_RAT | Somatostatin receptor | Somatostatin receptor type 4 | Sstr4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 42096.84 |
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| Organism: | RAT |
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| Description: | SOMATOSTATIN SST4 SSTR4 RAT::P30937 |
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| Residue: | 384 |
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| Sequence: | MNTPATLPLGGEDTTWTPGINASWAPDEEEDAVRSDGTGTAGMVTIQCIYALVCLVGLVG
NALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASAAALRHWPFGAVLCRAVLS
VDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAVF
ADTRPARGGEAVACNLHWPHPAWSAVFVIYTFLLGFLLPVLAIGLCYLLIVGKMRAVALR
AGWQQRRRSEKKITRLVLMVVTVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANS
CANPILYGFLSDNFRRSFQRVLCLRCCLLETTGGAEEEPLDYYATALKSRGGPGCICPPL
PCQQEPMQAEPACKRVPFTKTTTF
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| BDBM50065453 |
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| n/a |
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| Name | BDBM50065453 |
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| Synonyms: | (5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-dibenzyl-8-((R)-1-hydroxy-ethyl)-14-(1H-indol-3-ylmethyl)-tetradecahydro-3a,6,9,12,15,18-hexaaza-cyclopentacyclooctadecene-4,7,10,13,16,19-hexaone | CHEMBL421362 | L-361,301 | L-363,301 | L-363301 |
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| Type | Small organic molecule |
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| Emp. Form. | C44H54N8O7 |
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| Mol. Mass. | 806.949 |
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| SMILES | C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O |
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| Structure | 
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