| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Basic phospholipase A2 VRV-PL-VIIIa |
|---|
| Ligand | BDBM50242996 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_1672475 |
|---|
| IC50 | 24142±n/a nM |
|---|
| Citation |  Lokeshwari, DM; Rekha, ND; Srinivasan, B; Vivek, HK; Kariyappa, AK Design, synthesis of novel furan appended benzothiazepine derivatives and in vitro biological evaluation as potent VRV-PL-8a and H Bioorg Med Chem Lett27:3048-3054 (2017) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Basic phospholipase A2 VRV-PL-VIIIa |
|---|
| Name: | Basic phospholipase A2 VRV-PL-VIIIa |
|---|
| Synonyms: | 3.1.1.4 | Basic phospholipase A2 VRV-PL-VIIIa | DPLA2 | PA2B8_DABRR | PLA24 | Phosphatidylcholine 2-acylhydrolase | Phospholipase A2 4 | svPLA2 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 13615.14 |
|---|
| Organism: | Daboia russelii |
|---|
| Description: | ChEMBL_116772 |
|---|
| Residue: | 121 |
|---|
| Sequence: | SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPK
SDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELK
C
|
|
|
|---|
| BDBM50242996 |
|---|
| n/a |
|---|
| Name | BDBM50242996 |
|---|
| Synonyms: | CHEMBL4062876 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H14BrNOS |
|---|
| Mol. Mass. | 384.29 |
|---|
| SMILES | Brc1ccc(cc1)C1CC(=Nc2ccccc2S1)c1ccco1 |c:10| |
|---|
| Structure | 
|
|---|
Search and Browse
