| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor |
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| Ligand | BDBM50004665 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_138302 |
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| Kd | 1200±n/a nM |
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| Citation |  Nilsson, BM; Vargas, HM; Hacksell, U Urea and 2-imidazolidone derivatives of the muscarinic agents oxotremorine and N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide. J Med Chem35:3270-9 (1992) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Muscarinic acetylcholine receptor |
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| Name: | Muscarinic acetylcholine receptor |
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| Synonyms: | GPM3 | Muscarinic acetylcholine receptor M3 |
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| Type: | n/a |
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| Mol. Mass.: | 66272.13 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 587 |
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| Sequence: | MTLHSNSTTLPLFPNISTSWIHSPSEAGLPPGTVTHFGSYNISQAAGNFSSLNGTTSDPL
GGHTIWQVVFIAFLTGFLALVTIIGNILVIVSFKVNKQLKHVNNYFLLSLADLIIGVISM
NLFTTYIIMNRWALGNLACDLWLSIDYVASNASVMNLLVISFDRYFSITRPLTYRAKRTT
KRAGVMIGLAWVISFVLWAPAILFWQYFVGKRTVPPGECFIQFLSEPTITFGTAIAAFYM
PVTIMTILYWRIYKETEKRTKELAGLQASGTEAETENFVHPTGSSRSCSSYELQQQSLKH
SSRRKYSRCHFWFATKSWKPNAGQMDQDHSSSDSWNNYDAAASLENSASDEEDIGSETRA
IYSIVLKLPGHSTILNSTKLPSSDNLQVPEEDLEPMDMERNASKPQTQKSMDDGGSFQKS
FSNLPIQLESTMDTAKTSDANSSVSKTMATLPLSFKEATLAKRFALRTRSQITKRKRMSL
IKEKRAAQTLSAILLAFIITWTPYNIMVLVNTFCDSCIPKTYWNLGYWLCYINSTVNPVC
YALCNKTFRNTFKMLLLCQCDKRKRRKQQYQQRQSVIFHKRVPEQAL
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| BDBM50004665 |
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| n/a |
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| Name | BDBM50004665 |
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| Synonyms: | (oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | 1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | 1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one (oxotremorphine) | 1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one(Oxotremorine) | 1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidinium | CHEMBL7634 | Oxotremorine | Oxotremorine1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | cid_4630 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H18N2O |
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| Mol. Mass. | 206.2841 |
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| SMILES | O=C1CCCN1CC#CCN1CCCC1 |
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| Structure | 
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