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TargetSignal transduction protein TRAP
LigandBDBM50260007
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1692280 (CHEMBL4042929)
EC50 11400±n/a nM
Citation Vermote, ABrackman, GRisseeuw, MDCappoen, DCos, PCoenye, TVan Calenbergh, S Novel Potentiators for Vancomycin in the Treatment of Biofilm-Related MRSA Infections via a Mix and Match Approach. ACS Med Chem Lett8:38-42 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Signal transduction protein TRAP
Name:Signal transduction protein TRAP
Synonyms:Signal transduction protein TRAP | TRAP_STAAM | Target of RNAIII-activating protein | traP
Type:PROTEIN
Mol. Mass.:19547.99
Organism:Staphylococcus aureus (strain Mu50 / ATCC 700699)
Description:ChEMBL_117552
Residue:167
Sequence:
MKKLYTSYGTYGFLHQIKINNPTHQLFQFSASDTSVIFEETDGETVLKSPSIYEVIKEIG
EFSEHHFYCAIFIPSTEDHAYQLEKKLISVDDNFRNFGGFKSYRLLRPAKGTTYKIYFGF
ADRHAYEDFKQSDAFNDHFSKDALSHYFGSSGQHSSYFERYLYPIKE
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BDBM50260007
n/a
NameBDBM50260007
Synonyms:CHEMBL4102095
TypeSmall organic molecule
Emp. Form.C19H18N4O6
Mol. Mass.398.3694
SMILESO[C@@H]1[C@@H](CN2C(=O)c3ccccc3C2=O)OC[C@@]1(O)CNC(=O)c1ccnnc1 |r|
Structure
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