Reaction Details |
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Target | G-protein coupled receptor 55 |
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Ligand | BDBM50269024 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_1705585 (CHEMBL4056818) |
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EC50 | 300±n/a nM |
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Citation | Fakhouri, L; Cook, CD; Al-Huniti, MH; Console-Bram, LM; Hurst, DP; Spano, MBS; Nasrallah, DJ; Caron, MG; Barak, LS; Reggio, PH; Abood, ME; Croatt, MP Design, synthesis and biological evaluation of GPR55 agonists. Bioorg Med Chem25:4355-4367 (2017) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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G-protein coupled receptor 55 |
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Name: | G-protein coupled receptor 55 |
Synonyms: | G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN |
Type: | PROTEIN |
Mol. Mass.: | 36649.72 |
Organism: | Homo sapiens (Human) |
Description: | ChEMBL_1292265 |
Residue: | 319 |
Sequence: | MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
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BDBM50269024 |
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n/a |
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Name | BDBM50269024 |
Synonyms: | CHEMBL4060069 |
Type | Small organic molecule |
Emp. Form. | C27H25N3O4S2 |
Mol. Mass. | 519.635 |
SMILES | CN(c1ccccc1)S(=O)(=O)c1ccc(NC(=S)NC(=O)c2ccc3cc(CCO)ccc3c2)cc1 |
Structure |
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