| Reaction Details |
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 | Report a problem with these data |
| Target | D(2) dopamine receptor |
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| Ligand | BDBM50019878 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_62569 (CHEMBL671500) |
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| Ki | 280±n/a nM |
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| Citation |  Harrold, MW; Chang, YA; Wallace, RA; Farooqui, T; Wallace, LJ; Uretsky, N; Miller, DD Charged analogues of chlorpromazine as dopamine antagonists. J Med Chem30:1631-5 (1987) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| D(2) dopamine receptor |
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| Name: | D(2) dopamine receptor |
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| Synonyms: | DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2_RAT | Dopamine D2 receptor | Dopamine2-like | Drd2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 50931.60 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | P61169 |
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| Residue: | 444 |
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| Sequence: | MDPLNLSWYDDDLERQNWSRPFNGSEGKADRPHYNYYAMLLTLLIFIIVFGNVLVCMAVS
REKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTA
SILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPLLFGLNNTDQN
ECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRKRRKRVNTKRSSRAFRANLKTPL
KGNCTHPEDMKLCTVIMKSNGSFPVNRRRMDAARRAQELEMEMLSSTSPPERTRYSPIPP
SHHQLTLPDPSHHGLHSNPDSPAKPEKNGHAKIVNPRIAKFFEIQTMPNGKTRTSLKTMS
RRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNS
AVNPIIYTTFNIEFRKAFMKILHC
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| BDBM50019878 |
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| n/a |
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| Name | BDBM50019878 |
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| Synonyms: | CHEMBL44394 | [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-sulfonium; iodide |
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| Type | Small organic molecule |
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| Emp. Form. | C17H19ClNS2 |
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| Mol. Mass. | 336.922 |
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| SMILES | C[S+](C)CCCN1c2ccccc2Sc2ccc(Cl)cc12 |
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| Structure | 
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