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TargetCytosol aminopeptidase [33-68,L62W]
LigandBDBM50457473
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1759783 (CHEMBL4194791)
IC50 30±n/a nM
Citation Amin, SAAdhikari, NJha, T Design of Aminopeptidase N Inhibitors as Anti-cancer Agents. J Med Chem61:6468-6490 (2018) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cytosol aminopeptidase [33-68,L62W]
Name:Cytosol aminopeptidase [33-68,L62W]
Synonyms:AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP)
Type:Enzyme
Mol. Mass.:4015.44
Organism:Sus scrofa (Pig)
Description:P28839[33-68,L62W]
Residue:36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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  Blast E-value cutoff:
BDBM50457473
n/a
NameBDBM50457473
Synonyms:CHEMBL4209822
TypeSmall organic molecule
Emp. Form.C16H22N2O6
Mol. Mass.338.3557
SMILESCC(C)C[C@@H]([C@H](O)C(=O)NO)C(=O)N[C@H](C(O)=O)c1ccccc1 |r|
Structure
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