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TargetPhenylethanolamine N-methyltransferase
LigandBDBM50023170
Substrate/Competitorn/a
Meas. Tech.ChEBML_153310
Ki 4140±n/a nM
Citation Grunewald, GLCarter, AESall, DJMonn, JA Conformational preference for the binding of biaryl substrates and inhibitors to the active site of phenylethanolamine N-methyltransferase. J Med Chem31:60-5 (1988) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Phenylethanolamine N-methyltransferase
Name:Phenylethanolamine N-methyltransferase
Synonyms:Noradrenaline N-methyltransferase | PNMT | PNMT_BOVIN | PNMTase
Type:Enzyme
Mol. Mass.:30916.97
Organism:Bos taurus (bovine)
Description:n/a
Residue:283
Sequence:
MSGTDRSQAAGAVPDSDPGLAAVSSAYQRFEPRAYLRNNYAPPRGDLSCPDGVGPWKLRC
LAQTFATGEVSGRTLIDIGSGPTIYQLLSACAHFEDITMTDFLEVNRQELRLWLREEPGA
FDWSVYSQHVCLIEGKGESWQEKECQLRARVKRILPIDVHRPQPLGAGGLAPLPADALVS
AFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLAVVPVREEEVR
EALVRTATRCGICARTPMPAHLQTGVDDVKGIFFTRAQKKVGV
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  Blast E-value cutoff:
BDBM50023170
n/a
NameBDBM50023170
Synonyms:1-(9H-Fluoren-1-yl)-ethylamine | CHEMBL350036
TypeSmall organic molecule
Emp. Form.C15H15N
Mol. Mass.209.2863
SMILESCC(N)c1cccc-2c1Cc1ccccc-21
Structure
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