| Reaction Details |
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 | Report a problem with these data |
| Target | Integrase |
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| Ligand | BDBM50484860 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_809660 (CHEMBL2015879) |
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| IC50 | 52±n/a nM |
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| Citation |  Agapkina, J; Zatsepin, T; Knyazhanskaya, E; Mouscadet, JF; Gottikh, M Structure-Activity Relationship Studies of HIV-1 Integrase Oligonucleotide Inhibitors. ACS Med Chem Lett2:532-7 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Integrase |
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| Name: | Integrase |
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| Synonyms: | pol |
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| Type: | PROTEIN |
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| Mol. Mass.: | 32203.43 |
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| Organism: | Human immunodeficiency virus 1 |
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| Description: | ChEMBL_106649 |
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| Residue: | 288 |
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| Sequence: | FLDGIDKAQEEHEKYHSNWRAMASDFNLPPVVAKEIVASCDKCQLKGEAMHGQVDCSPGI
WQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSN
FTSTTVKAACWWAGIKQEFGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAV
FIHNFKRKGGIGGYSAGERIVDIIATDIQTKELQKQITKIQNFRVYYRDSRDPVWKGPAK
LLWKGEGAVVIQDNSDIKVVPRRKAKIIRDYGKQMAGDDCVASRQDED
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| BDBM50484860 |
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| n/a |
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| Name | BDBM50484860 |
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| Synonyms: | CHEMBL2012379 |
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| Type | Small organic molecule |
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| Emp. Form. | C141H166Cl6N35O91P11 |
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| Mol. Mass. | 4360.436 |
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| SMILES | n/a |
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| Structure | 
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