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TargetSolute carrier family 22 member 8
LigandBDBM50206509
Substrate/Competitorn/a
Meas. Tech.ChEMBL_836315 (CHEMBL2076479)
Ki 4430±n/a nM
Citation Nagata, YKusuhara, HEndou, HSugiyama, Y Expression and functional characterization of rat organic anion transporter 3 (rOat3) in the choroid plexus. Mol Pharmacol61:982-8 (2002) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Solute carrier family 22 member 8
Name:Solute carrier family 22 member 8
Synonyms:Oat3 | Organic anion transporter 3 | S22A8_RAT | Slc22a8 | rOat3
Type:PROTEIN
Mol. Mass.:59199.83
Organism:Rattus norvegicus
Description:ChEMBL_1482580
Residue:536
Sequence:
MTFSEILDRVGSMGPFQYLHVTLLALPVLGIANHNLLQIFTATTPVHHCRPPPNASIGPW
VLPLDPNGKPEKCLRFVHLPNASLPNDTQRATEPCLDGWIYNSTRDTIVIEWDLVCSSNK
LKEMAQSIFMAGILVGGPVIGELSDRFGRKPILTWSYLMLAASGSGAAFSPSLPVYMIFR
FLCGCSISGISLSTVILNVEWVPTSMRAISSTSIGYCYTIGQFILSGLAYAIPQWRWLQL
TSSAPFFIFSLLSWWVPESIRWLVLSGKYSKALKTLQRVATFNGKKEEGKKLTIEELKFN
LQKDITSAKVKYGLSDLFRVSILRRVTFCLSLAWFSTGFAYYSLAMGVEEFGVNIYILQI
IFGGVDIPAKFITILSLSYLGRRITQSFLLLLAGGAILALIFVPSEMQLLRTALAVFGKG
CLSGSFSCLFLYTSELYPTVLRQTGMGISNVWARVGSMIAPLVKITGELQPFIPNVIFGT
TALLGGSAAFFLLETLNRPLPETIEDIQNWHKQVQKTKQESEAEKASQIIPLKTGG
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50206509
n/a
NameBDBM50206509
Synonyms:4-Dipropylsulfamoyl-benzoic acid | 4-Dipropylsulfamoyl-benzoic acid anion | 4-Dipropylsulfamoyl-benzoic acid(probenecid) | Benemid | CHEMBL897 | PROBENECID | Probalan
TypeSmall organic molecule
Emp. Form.C13H19NO4S
Mol. Mass.285.359
SMILESCCCN(CCC)S(=O)(=O)c1ccc(cc1)C(O)=O
Structure
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