| Reaction Details |
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 | Report a problem with these data |
| Target | Solute carrier organic anion transporter family member 1A1 |
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| Ligand | BDBM50375594 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_837108 (CHEMBL2076360) |
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| Ki | 32000±n/a nM |
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| Citation |  Pang, KS; Wang, PJ; Chung, AY; Wolkoff, AW The modified dipeptide, enalapril, an angiotensin-converting enzyme inhibitor, is transported by the rat liver organic anion transport protein. Hepatology28:1341-6 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Solute carrier organic anion transporter family member 1A1 |
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| Name: | Solute carrier organic anion transporter family member 1A1 |
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| Synonyms: | OATP-1 | Oatp1 | Oatp1a1 | Organic anion-transporting polypeptide 1 | SO1A1_RAT | Slc21a1 | Slco1a1 | Sodium-independent organic anion transporter 1 | Solute carrier family 21 member 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 74188.94 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_838286 |
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| Residue: | 670 |
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| Sequence: | MEETEKKIATQEGRLFSKMKVFLLSLTCACLTKSLSGVYMNSMLTQIERQFDISTSVAGL
INGSFEIGNLFFIVFVSYFGTKLHRPVVIGIGCVIMGLGCLLMSLPHFFMGRYEYETTIS
PTGNLSSNSFLCMENRTQTLKPTQDPAECVKEMKSLMWICVMVGNIIRGIGETPIVPLGI
SYIEDFAKSENSPLYIGILEMGKVAGPIFGLLLGSYCAQIYVDIGSVNTDDLTITPSDTR
WVGAWWIGFLVCAGVNILTSIPFFFLPKALPKKGQQENVAVTKDGKVEKYGGQAREENLG
ITKDFLTFMKRLFCNPIYMLFILTSVLQVNGFINKFTFLPKYLEQQYGKSTAEAIFLIGV
YSLPPICLGYLIGGFIMKKFKITVKKAAYLAFCLSVFEYLLFLCHFMLTCDNAAVAGLTT
SYKGVQHQLHVESKVLADCNTRCSCSTNTWDPVCGDNGVAYMSACLAGCKKFVGTGTNMV
FQDCSCIQSLGNSSAVLGLCKKGPECANRLQYFLILTIIISFIYSLTAIPGYMVFLRCVK
SEEKSLGVGLHTFCIRVFAGIPAPVYFGALIDRTCLHWGTLKCGQRGACRMYDINSFRHI
YLGLPIALRGSSYLPAFFILILMRKFQFPGDIDSSATDHTEMMLGEKESEHTDVHGSPQV
ENDGELKTKL
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| BDBM50375594 |
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| n/a |
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| Name | BDBM50375594 |
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| Synonyms: | TAUROCHOLATE |
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| Type | Small organic molecule |
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| Emp. Form. | C26H45NO7S |
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| Mol. Mass. | 515.703 |
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| SMILES | C[C@H](CCC(=O)NCCS(O)(=O)=O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C |r| |
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| Structure | 
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