| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Solute carrier family 15 member 2 |
|---|
| Ligand | BDBM84007 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_836935 (CHEMBL2075775) |
|---|
| IC50 | 3200000±n/a nM |
|---|
| Citation |  Ganapathy, ME; Prasad, PD; Mackenzie, B; Ganapathy, V; Leibach, FH Interaction of anionic cephalosporins with the intestinal and renal peptide transporters PEPT 1 and PEPT 2. Biochim Biophys Acta1324:296-308 (1997) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Solute carrier family 15 member 2 |
|---|
| Name: | Solute carrier family 15 member 2 |
|---|
| Synonyms: | Oligopeptide transporter, kidney isoform | Pept2 | S15A2_RAT | Slc15a2 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 81331.63 |
|---|
| Organism: | Rattus norvegicus |
|---|
| Description: | ChEMBL_838253 |
|---|
| Residue: | 729 |
|---|
| Sequence: | MNPFQKNESKETLFSPVSTEEMLPRPPSPPKKSPPKIFGSSYPVSIAFIVVNEFCERFSY
YGMKAVLTLYFLYFLHWNEDTSTSVYHAFSSLCYFTPILGAAIADSWLGKFKTIIYLSLV
YVLGHVFKSLGAIPILGGKMLHTILSLVGLSLIALGTGGIKPCVAAFGGDQFEEEHAEAR
TRYFSVFYLAINAGSLISTFITPMLRGDVKCFGQDCYALAFGVPGLLMVLALVVFAMGSK
MYRKPPPEGNIVAQVIKCIWFALCNRFRNRSGDLPKRQHWLDWAAEKYPKHLIADVKALT
RVLFLYIPLPMFWALLDQQGSRWTLQANKMNGDLGFFVLQPDQMQVLNPFLVLIFIPLFD
LVIYRLISKCRINFSSLRKMAVGMILACLAFAVAALVETKINGMIHPQPASQEIFLQVLN
LADGDVKVTVLGSRNNSLLVESVSSFQNTTHYSKLHLEAKSQDLHFHLKYNSLSVHNDHS
VEEKNCYQLLIHQDGESISSMLVKDTGIKPANGMAAIRFINTLHKDLNISLDTDAPLSVG
KDYGVSAYRTVLRGKYPAVHCETEDKVFSLDLGQLDFGTTYLFVITNITSQGLQAWKAED
IPVNKLSIAWQLPQYVLVTAAEVMFSVTGLEFSYSQAPSSMKSVLQAAWLLTVAVGNIIV
LVVAQFSGLAQWAEFVLFSCLLLVVCLIFSVMAYYYVPLKSEDTREATDKQIPAVQGNMI
NLETKNTRL
|
|
|
|---|
| BDBM84007 |
|---|
| n/a |
|---|
| Name | BDBM84007 |
|---|
| Synonyms: | CEFIXIME | Cefiximum [Latin] | MLS002222332 | SMR001307271 | cid_5362065 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H15N5O7S2 |
|---|
| Mol. Mass. | 453.45 |
|---|
| SMILES | Nc1nc(cs1)C(=N\OCC(O)=O)\C(=O)N[C@H]1[C@H]2SCC(C=C)=C(N2C1=O)C(O)=O |c:23| |
|---|
| Structure | 
|
|---|
Search and Browse
