| Reaction Details |
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 | Report a problem with these data |
| Target | Serine protease 1 |
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| Ligand | BDBM50031251 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_213087 (CHEMBL815015) |
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| Ki | 20900±n/a nM |
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| Citation |  Angliker, H Synthesis of tight binding inhibitors and their action on the proprotein-processing enzyme furin. J Med Chem38:4014-8 (1995) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Serine protease 1 |
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| Name: | Serine protease 1 |
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| Synonyms: | Alpha-trypsin chain 1 | Alpha-trypsin chain 2 | Beta-trypsin | Cationic trypsinogen | PRSS1 | Serine protease 1 | TRP1 | TRY1 | TRY1_HUMAN | TRYP1 | Thrombin & trypsin | Trypsin | Trypsin I | Trypsin-1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 26557.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P07477 |
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| Residue: | 247 |
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| Sequence: | MNPLLILTFVAAALAAPFDDDDKIVGGYNCEENSVPYQVSLNSGYHFCGGSLINEQWVVS
AGHCYKSRIQVRLGEHNIEVLEGNEQFINAAKIIRHPQYDRKTLNNDIMLIKLSSRAVIN
ARVSTISLPTAPPATGTKCLISGWGNTASSGADYPDELQCLDAPVLSQAKCEASYPGKIT
SNMFCVGFLEGGKDSCQGDSGGPVVCNGQLQGVVSWGDGCAQKNKPGVYTKVYNYVKWIK
NTIAANS
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| BDBM50031251 |
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| n/a |
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| Name | BDBM50031251 |
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| Synonyms: | (R)-2-{2-[(R)-2-((S)-5-{(S)-6-Amino-2-[(S)-2-((S)-2-decylamino-5-guanidino-pentanoylamino)-3-methyl-butyrylamino]-hexanoylamino}-8-guanidino-4-oxo-octanoylamino)-3-methyl-butyrylamino]-acetylamino}-4-methyl-pentanoic acid methyl ester | CHEMBL410994 |
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| Type | Small organic molecule |
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| Emp. Form. | C50H96N14O9 |
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| Mol. Mass. | 1037.3856 |
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| SMILES | CCCCCCCCCCN[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)CCC(=O)N[C@H](C(C)C)C(=O)NCC(=O)N[C@H](CC(C)C)C(=O)OC |
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| Structure | 
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