| Reaction Details |
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 | Report a problem with these data |
| Target | Voltage-dependent L-type calcium channel subunit alpha-1C |
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| Ligand | BDBM50487586 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_910383 (CHEMBL3056066) |
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| IC50 | 1.7±n/a nM |
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| Citation |  TBA Med Chem Res19:58-70 (2010) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Voltage-dependent L-type calcium channel subunit alpha-1C |
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| Name: | Voltage-dependent L-type calcium channel subunit alpha-1C |
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| Synonyms: | CAC1C_CAVPO | CACH2 | CACH2 | CACN2 | CACNA1C | CACNL1A1 | CCHL1A1 | Calcium channel, L type, alpha-1 polypeptide, isoform 1, cardiac muscle | Voltage-dependent L-type calcium channel subunit alpha-1C | Voltage-gated calcium channel subunit alpha Cav1.2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 19518.62 |
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| Organism: | Cavia porcellus |
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| Description: | ChEMBL_106600 |
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| Residue: | 169 |
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| Sequence: | FQEQGEQEYKNCELDKNQRQCVEYALKARPLRRYIPISITFFRLFRVMRLVKLLSRGEGI
RTLLWTFIKSFQALPYVALLIVMLFFIYAVIGMQVFGKIALNDTTEINRNNNFQTFPQAV
LLLFRCATGEAWQDIMLACMPGKKRAPESEPSNSTEGETPCGSSFAVFY
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| BDBM50487586 |
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| n/a |
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| Name | BDBM50487586 |
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| Synonyms: | CHEMBL2261194 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H24ClN3O4 |
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| Mol. Mass. | 429.897 |
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| SMILES | CCc1nc(Cl)c([nH]1)C1C(C(=O)OC)=C(C)NC(C)=C1C(=O)OCc1ccccc1 |c:19,t:14| |
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| Structure | 
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