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TargetCasein kinase 1, delta tv1
LigandBDBM50488802
Substrate/Competitorn/a
Meas. Tech.ChEMBL_932131 (CHEMBL3072203)
IC50 410±n/a nM
Citation  TBA Med Chem Res22:3247-3258 (2013)    Article
More Info.:Get all data from this article,  Assay Method
 
Casein kinase 1, delta tv1
Name:Casein kinase 1, delta tv1
Synonyms:CSNK1D
Type:PROTEIN
Mol. Mass.:47258.61
Organism:Sus scrofa
Description:ChEMBL_106594
Residue:415
Sequence:
MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQ
GGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIH
SKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYA
SINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVL
CKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRA
ADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEAAPPTPLTPTSHTANTSPRPV
SGMERERKVSMRLHRGAPVNISSSDLTGRQDTSRMSTSQIAGRVAASGLQSAVHR
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  Blast E-value cutoff:
BDBM50488802
n/a
NameBDBM50488802
Synonyms:CHEMBL2295951
TypeSmall organic molecule
Emp. Form.C18H16ClN7
Mol. Mass.365.82
SMILESCC(C)n1cnc2c(Nc3ccc(cc3)-c3cncnc3)nc(Cl)nc12
Structure
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