| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor |
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| Ligand | BDBM50036163 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_138314 (CHEMBL743825) |
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| Ki | 1300±n/a nM |
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| Citation |  Nilsson, BM; Sundquist, S; Johansson, G; Nordvall, G; Glas, G; Nilvebrant, L; Hacksell, U 3-Heteroaryl-substituted quinuclidin-3-ol and quinuclidin-2-ene derivatives as muscarinic antagonists. Synthesis and structure-activity relationships. J Med Chem38:473-87 (1995) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Muscarinic acetylcholine receptor |
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| Name: | Muscarinic acetylcholine receptor |
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| Synonyms: | GPM3 | Muscarinic acetylcholine receptor M3 |
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| Type: | n/a |
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| Mol. Mass.: | 66272.13 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 587 |
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| Sequence: | MTLHSNSTTLPLFPNISTSWIHSPSEAGLPPGTVTHFGSYNISQAAGNFSSLNGTTSDPL
GGHTIWQVVFIAFLTGFLALVTIIGNILVIVSFKVNKQLKHVNNYFLLSLADLIIGVISM
NLFTTYIIMNRWALGNLACDLWLSIDYVASNASVMNLLVISFDRYFSITRPLTYRAKRTT
KRAGVMIGLAWVISFVLWAPAILFWQYFVGKRTVPPGECFIQFLSEPTITFGTAIAAFYM
PVTIMTILYWRIYKETEKRTKELAGLQASGTEAETENFVHPTGSSRSCSSYELQQQSLKH
SSRRKYSRCHFWFATKSWKPNAGQMDQDHSSSDSWNNYDAAASLENSASDEEDIGSETRA
IYSIVLKLPGHSTILNSTKLPSSDNLQVPEEDLEPMDMERNASKPQTQKSMDDGGSFQKS
FSNLPIQLESTMDTAKTSDANSSVSKTMATLPLSFKEATLAKRFALRTRSQITKRKRMSL
IKEKRAAQTLSAILLAFIITWTPYNIMVLVNTFCDSCIPKTYWNLGYWLCYINSTVNPVC
YALCNKTFRNTFKMLLLCQCDKRKRRKQQYQQRQSVIFHKRVPEQAL
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|
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| BDBM50036163 |
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| n/a |
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| Name | BDBM50036163 |
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| Synonyms: | 3-Benzofuran-2-yl-1-methyl-1-azonia-bicyclo[2.2.2]oct-2-ene | CHEMBL144435 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H18NO |
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| Mol. Mass. | 240.3197 |
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| SMILES | n/a |
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| Structure | 
|
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