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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50041255
Substrate/Competitorn/a
Meas. Tech.ChEMBL_200976 (CHEMBL802063)
Ki 0.38±n/a nM
Citation Glennon, RAAblordeppey, SYIsmaiel, AMel-Ashmawy, MBFischer, JBHowie, KB Structural features important for sigma 1 receptor binding. J Med Chem37:1214-9 (1994) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:Aging-associated gene 8 protein | OPRS1 | SGMR1_HUMAN | SIG-1R | SIGMAR1 | SR-BP | SR31747-binding protein | SRBP | Sigma 1-type opioid receptor | Sigma opioid receptor | Sigma1R | hSigmaR1
Type:Enzyme Catalytic Domain
Mol. Mass.:25124.85
Organism:Homo sapiens (Human)
Description:Q99720
Residue:223
Sequence:
MQWAVGRRWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLFGQDP
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  Blast E-value cutoff:
BDBM50041255
n/a
NameBDBM50041255
Synonyms:CHEMBL19637 | Methyl-(5-phenyl-pentyl)-(3-phenyl-propyl)-amine
TypeSmall organic molecule
Emp. Form.C21H29N
Mol. Mass.295.4617
SMILESCN(CCCCCc1ccccc1)CCCc1ccccc1
Structure
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