| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma non-opioid intracellular receptor 1 |
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| Ligand | BDBM81924 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_201887 (CHEMBL809042) |
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| IC50 | 430±n/a nM |
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| Citation |  Sonesson, C; Waters, N; Svensson, K; Carlsson, A; Smith, MW; Piercey, MF; Meier, E; Wikström, H Substituted 3-phenylpiperidines: new centrally acting dopamine autoreceptor antagonists. J Med Chem36:3188-96 (1993) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Sigma non-opioid intracellular receptor 1 |
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| Name: | Sigma non-opioid intracellular receptor 1 |
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| Synonyms: | Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 25266.54 |
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| Organism: | RAT |
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| Description: | Q9R0C9 |
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| Residue: | 223 |
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| Sequence: | MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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| BDBM81924 |
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| n/a |
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| Name | BDBM81924 |
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| Synonyms: | (R)-3-(1-Propyl-piperidin-3-yl)-phenol | 3PPP(+/-) | CAS_85976-54-1 | CHEMBL276500 | NSC_202477 | PPP, R(+)-3 | PPP, S(-)-3 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H21NO |
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| Mol. Mass. | 219.3226 |
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| SMILES | CCCN1CCCC(C1)c1cccc(O)c1 |
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| Structure | 
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