| Reaction Details |
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 | Report a problem with these data |
| Target | Acyl-protein thioesterase 1 |
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| Ligand | BDBM207992 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1300899 (CHEMBL3135186) |
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| Ki | >10000±n/a nM |
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| Citation |  Davda, D; Martin, BR Acyl protein thioesterase inhibitors as probes of dynamic S-palmitoylation. Medchemcomm5:268-276 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Acyl-protein thioesterase 1 |
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| Name: | Acyl-protein thioesterase 1 |
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| Synonyms: | APT-1 | APT1 | Acyl-protein thioesterase 1 (APT1 WT) | LPL-I | LPL1 | LYPA1_HUMAN | LYPLA1 | LysoPLA I | Lysophospholipase 1 | Lysophospholipase I | hAPT1 |
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| Type: | Protein |
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| Mol. Mass.: | 24670.33 |
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| Organism: | Homo sapiens (Human) |
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| Description: | O75608 |
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| Residue: | 230 |
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| Sequence: | MCGNNMSTPLPAIVPAARKATAAVIFLHGLGDTGHGWAEAFAGIRSSHIKYICPHAPVRP
VTLNMNVAMPSWFDIIGLSPDSQEDESGIKQAAENIKALIDQEVKNGIPSNRIILGGFSQ
GGALSLYTALTTQQKLAGVTALSCWLPLRASFPQGPIGGANRDISILQCHGDCDPLVPLM
FGSLTVEKLKTLVNPANVTFKTYEGMMHSSCQQEMMDVKQFIDKLLPPID
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| BDBM207992 |
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| n/a |
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| Name | BDBM207992 |
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| Synonyms: | ML349 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H22N2O4S2 |
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| Mol. Mass. | 454.562 |
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| SMILES | COc1ccc(cc1)N1CCN(CC1)C(=O)c1cc2CS(=O)(=O)c3ccccc3-c2s1 |
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| Structure | 
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