| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 4 |
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| Ligand | BDBM50058170 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_3347 (CHEMBL619047) |
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| Ki | 1.05±n/a nM |
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| Citation |  Soulier, JL; Yang, D; Brémont, B; Croci, T; Guzzi, U; Langlois, M Arylcarbamate derivatives of 1-piperidineethanol as potent ligands for 5-HT4 receptors. J Med Chem40:1755-61 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| 5-hydroxytryptamine receptor 4 |
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| Name: | 5-hydroxytryptamine receptor 4 |
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| Synonyms: | 5-HT-4 | 5-HT4 | 5-HT4L | 5-HT4S | 5-hydroxytryptamine receptor 4 | 5HT4R_RAT | Htr4 | Serotonin (5-HT) receptor | Serotonin 4 (5-HT4) receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 46117.31 |
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| Organism: | RAT |
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| Description: | 5-HT4 HTR4 RAT::Q62758 |
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| Residue: | 406 |
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| Sequence: | MDRLDANVSSNEGFGSVEKVVLLTFFAMVILMAILGNLLVMVAVCRDRQLRKIKTNYFIV
SLAFADLLVSVLVNAFGAIELVQDIWFYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYY
AICCQPLVYRNKMTPLRIALMLGGCWVIPMFISFLPIMQGWNNIGIVDVIEKRKFNHNSN
STFCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAQQIQMLQRAGATSESRP
QTADQHSTHRMRTETKAAKTLCVIMGCFCFCWAPFFVTNIVDPFIDYTVPEKVWTAFLWL
GYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYKRPPILGQTVPCSTTTINGSTHVLRD
TVECGGQWESRCHLTATSPLVAAQPVIRRPQDNDLEDSCSLKRSQS
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| BDBM50058170 |
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| n/a |
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| Name | BDBM50058170 |
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| Synonyms: | (2-Ethoxy-phenyl)-carbamic acid 2-((3R,5S)-3,5-dimethyl-piperidin-1-yl)-ethyl ester | (2-Ethoxy-phenyl)-carbamic acid 2-((3S,5R)-3,5-dimethyl-piperidin-1-yl)-ethyl ester | CHEMBL48836 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H28N2O3 |
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| Mol. Mass. | 320.4265 |
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| SMILES | CCOc1ccccc1NC(=O)OCCN1C[C@@H](C)C[C@@H](C)C1 |
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| Structure | 
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