| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50059367 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_75462 (CHEMBL686360) |
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| IC50 | 4.5±n/a nM |
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| Citation |  Bryant, SD; Guerrini, R; Salvadori, S; Bianchi, C; Tomatis, R; Attila, M; Lazarus, LH Helix-inducing alpha-aminoisobutyric acid in opioid mimetic deltorphin C analogues. J Med Chem40:2579-87 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50059367 |
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| n/a |
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| Name | BDBM50059367 |
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| Synonyms: | (S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-2-methyl-propionylamino]-N-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propyl]-3-methyl-butyramide | CHEMBL420606 |
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| Type | Small organic molecule |
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| Emp. Form. | C37H54N8O8 |
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| Mol. Mass. | 738.8735 |
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| SMILES | CC(C)[C@H](NC(=O)[C@@H](NC(=O)C(C)(C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(=O)NCC(N)=O |
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| Structure | 
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