| Reaction Details |
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 | Report a problem with these data |
| Target | Beta-2 adrenergic receptor |
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| Ligand | BDBM50064207 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_38607 (CHEMBL652290) |
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| IC50 | >10000±n/a nM |
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| Citation |  Blanc, M; Tamir, A; Aubriot, S; Michel, MC; Bouzoubaa, M; Leclerc, G; Demenge, P Synthesis and adrenergic activity of a new series of N-aryl dicyclopropyl ketone oxime ethers: SAR and stereochemical aspects. J Med Chem41:1613-8 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Beta-2 adrenergic receptor |
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| Name: | Beta-2 adrenergic receptor |
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| Synonyms: | ADRB2 | ADRB2_CANLF |
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| Type: | PROTEIN |
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| Mol. Mass.: | 46593.67 |
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| Organism: | Canis familiaris |
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| Description: | ChEMBL_56504 |
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| Residue: | 415 |
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| Sequence: | MGQPANRSVFLLAPNGSHAPDQGDSQERSEAWVVGMGIVMSLIVLAIVFGNVLVITAIAR
FERLQTVTNYFITSLACADLVMGLAVVPFGASHILMKMWTFGNFWCEFWTSIDVLCVTAS
IETLCVIAVDRYFAITSPFKYQSLLTKNKARVVILMVWIVSGLTSFLPIQMHWYRATHQE
AINCYAKETCCDFFTNQAYAIASSIVSFYLPLVVMVFVYSRVFQVAQRQLQKIDRSEGRF
HAQNLSQVEQDGRSGHGHRRSSKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQD
NLIPKEVYILLNWVGYVNSAFNPLIYCRSPDFRIAFQELLCLRRSSLKAYGNGYSNNSNS
RSDYAGEHSGCHLGQEKDSELLCEDPPGTEDRQGTVPSDSVDSQGRNCSTNDSLL
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| BDBM50064207 |
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| n/a |
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| Name | BDBM50064207 |
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| Synonyms: | CHEMBL40217 | Dicyclopropyl-methanone O-(2-hydroxy-3-p-tolylamino-propyl)-oxime |
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| Type | Small organic molecule |
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| Emp. Form. | C17H24N2O2 |
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| Mol. Mass. | 288.3847 |
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| SMILES | Cc1ccc(NCC(O)CON=C(C2CC2)C2CC2)cc1 |
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| Structure | 
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