| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 84 |
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| Ligand | BDBM50511001 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1843332 (CHEMBL4343759) |
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| Ki | 1.3±n/a nM |
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| Citation |  Köse, M; Pillaiyar, T; Namasivayam, V; De Filippo, E; Sylvester, K; Ulven, T; von Kügelgen, I; Müller, CE An Agonist Radioligand for the Proinflammatory Lipid-Activated G Protein-Coupled Receptor GPR84 Providing Structural Insights. J Med Chem63:2391-2410 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 84 |
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| Name: | G-protein coupled receptor 84 |
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| Synonyms: | EX33 | G-protein coupled receptor 84 | GPR84 | GPR84_HUMAN | Inflammation-related G-protein coupled receptor EX33 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 43726.73 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_116040 |
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| Residue: | 396 |
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| Sequence: | MWNSSDANFSCYHESVLGYRYVAVSWGVVVAVTGTVGNVLTLLALAIQPKLRTRFNLLIA
NLTLADLLYCTLLQPFSVDTYLHLHWRTGATFCRVFGLLLFASNSVSILTLCLIALGRYL
LIAHPKLFPQVFSAKGIVLALVSTWVVGVASFAPLWPIYILVPVVCTCSFDRIRGRPYTT
ILMGIYFVLGLSSVGIFYCLIHRQVKRAAQALDQYKLRQASIHSNHVARTDEAMPGRFQE
LDSRLASGGPSEGISSEPVSAATTQTLEGDSSEVGDQINSKRAKQMAEKSPPEASAKAQP
IKGARRAPDSSSEFGKVTRMCFAVFLCFALSYIPFLLLNILDARVQAPRVVHMLAANLTW
LNGCINPVLYAAMNRQFRQAYGSILKRGPRSFHRLH
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| BDBM50511001 |
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| n/a |
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| Name | BDBM50511001 |
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| Synonyms: | CHEMBL4439640 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H15N3O2 |
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| Mol. Mass. | 245.2771 |
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| SMILES | Cc1ccc(CCNc2cc(=O)[nH]c(=O)[nH]2)cc1 |
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| Structure | 
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