| Reaction Details |
|---|
 | Report a problem with these data |
| Target | G-protein coupled receptor 84 |
|---|
| Ligand | BDBM50180948 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1843327 (CHEMBL4343754) |
|---|
| EC50 | 3490±n/a nM |
|---|
| Citation |  Köse, M; Pillaiyar, T; Namasivayam, V; De Filippo, E; Sylvester, K; Ulven, T; von Kügelgen, I; Müller, CE An Agonist Radioligand for the Proinflammatory Lipid-Activated G Protein-Coupled Receptor GPR84 Providing Structural Insights. J Med Chem63:2391-2410 (2020) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| G-protein coupled receptor 84 |
|---|
| Name: | G-protein coupled receptor 84 |
|---|
| Synonyms: | EX33 | G-protein coupled receptor 84 | GPR84 | GPR84_HUMAN | Inflammation-related G-protein coupled receptor EX33 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 43726.73 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_116040 |
|---|
| Residue: | 396 |
|---|
| Sequence: | MWNSSDANFSCYHESVLGYRYVAVSWGVVVAVTGTVGNVLTLLALAIQPKLRTRFNLLIA
NLTLADLLYCTLLQPFSVDTYLHLHWRTGATFCRVFGLLLFASNSVSILTLCLIALGRYL
LIAHPKLFPQVFSAKGIVLALVSTWVVGVASFAPLWPIYILVPVVCTCSFDRIRGRPYTT
ILMGIYFVLGLSSVGIFYCLIHRQVKRAAQALDQYKLRQASIHSNHVARTDEAMPGRFQE
LDSRLASGGPSEGISSEPVSAATTQTLEGDSSEVGDQINSKRAKQMAEKSPPEASAKAQP
IKGARRAPDSSSEFGKVTRMCFAVFLCFALSYIPFLLLNILDARVQAPRVVHMLAANLTW
LNGCINPVLYAAMNRQFRQAYGSILKRGPRSFHRLH
|
|
|
|---|
| BDBM50180948 |
|---|
| n/a |
|---|
| Name | BDBM50180948 |
|---|
| Synonyms: | CHEBI:30805 | DODECANOATE | Dodecanoic Acid | Dodecanoic Acid Anion | Lauric Acid |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C12H24O2 |
|---|
| Mol. Mass. | 200.3178 |
|---|
| SMILES | CCCCCCCCCCCC(O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
