| Reaction Details |
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 | Report a problem with these data |
| Target | Chemerin-like receptor 1 |
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| Ligand | BDBM50517133 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1867369 (CHEMBL4368344) |
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| IC50 | 150±n/a nM |
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| Citation |  Imaizumi, T; Kobayashi, A; Otsubo, S; Komai, M; Magara, M; Otsubo, N The discovery and optimization of a series of 2-aminobenzoxazole derivatives as ChemR23 inhibitors. Bioorg Med Chem27:0 (2019) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Chemerin-like receptor 1 |
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| Name: | Chemerin-like receptor 1 |
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| Synonyms: | CML1_MOUSE | Chemokine-like receptor 1 | Cmklr1 | Dez | G-protein coupled receptor DEZ | Gpcr27 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41826.01 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_119019 |
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| Residue: | 371 |
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| Sequence: | MEYDAYNDSGIYDDEYSDGFGYFVDLEEASPWEAKVAPVFLVVIYSLVCFLGLLGNGLVI
VIATFKMKKTVNTVWFVNLAVADFLFNIFLPMHITYAAMDYHWVFGKAMCKISNFLLSHN
MYTSVFLLTVISFDRCISVLLPVWSQNHRSIRLAYMTCSAVWVLAFFLSSPSLVFRDTAN
IHGKITCFNNFSLAAPESSPHPAHSQVVSTGYSRHVAVTVTRFLCGFLIPVFIITACYLT
IVFKLQRNRLAKNKKPFKIIITIIITFFLCWCPYHTLYLLELHHTAVPSSVFSLGLPLAT
AVAIANSCMNPILYVFMGHDFRKFKVALFSRLANALSEDTGPSSYPSHRSFTKMSSLNEK
ASVNEKETSTL
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| BDBM50517133 |
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| n/a |
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| Name | BDBM50517133 |
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| Synonyms: | CHEMBL4448632 |
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| Type | Small organic molecule |
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| Emp. Form. | C28H29N7O2 |
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| Mol. Mass. | 495.5756 |
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| SMILES | CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2cc(ccc2o1)C(=O)NC |r| |
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| Structure | 
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