| Reaction Details |
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 | Report a problem with these data |
| Target | Casein kinase II subunit alpha 3 |
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| Ligand | BDBM50009001 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1869609 (CHEMBL4370675) |
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| IC50 | 10000±n/a nM |
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| Citation |  Zhao, L; Yuan, X; Wang, J; Feng, Y; Ji, F; Li, Z; Bian, J A review on flavones targeting serine/threonine protein kinases for potential anticancer drugs. Bioorg Med Chem27:677-685 (2019) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Casein kinase II subunit alpha 3 |
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| Name: | Casein kinase II subunit alpha 3 |
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| Synonyms: | 2.7.11.1 | CK II alpha 3 | CSK23_HUMAN | CSNK2A1P | CSNK2A3 | Casein kinase II alpha 1 polypeptide pseudogene | Casein kinase II subunit alpha 3 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 45229.76 |
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| Organism: | Homo sapiens |
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| Description: | ChEMBL_116899 |
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| Residue: | 391 |
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| Sequence: | MSGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINIT
NNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTD
FKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAE
FYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWRLGCMLASMIFRKEPFFHGRDNYD
QLVRIAKFLGTEDLYGYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDF
LDKLLRYDHQSRLTAREAMEHPYFYTVVKDQARMGSSSMPGGSTPVSSANVMSGISSVPT
PSPLGPLAGSPVIAAANPLGMPVPAATGAQQ
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| BDBM50009001 |
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| n/a |
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| Name | BDBM50009001 |
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| Synonyms: | 5,6,7-Trihydroxyflavone | 5,6,7-trihydroxy-2-phenyl-4H-chromen-4-one | Baicalein | Baicalein, 14 | Baicalein, 8 | CHEMBL8260 | US10252984, Table 2.33 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H10O5 |
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| Mol. Mass. | 270.2369 |
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| SMILES | Oc1cc2oc(cc(=O)c2c(O)c1O)-c1ccccc1 |
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| Structure | 
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