| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 1 |
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| Ligand | BDBM50065468 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_143836 (CHEMBL748719) |
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| IC50 | 1.7±n/a nM |
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| Citation |  Kordik, CP; Reitz, AB Pharmacological treatment of obesity: therapeutic strategies. J Med Chem42:181-201 (1999) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide Y receptor type 1 |
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| Name: | Neuropeptide Y receptor type 1 |
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| Synonyms: | FC5 | NPY-Y1 | NPY1-R | NPY1R_RAT | Neuropeptide Y receptor type 1 | Npy1r |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44126.41 |
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| Organism: | RAT |
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| Description: | NPY-Y1 NPY1R RAT::P21555 |
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| Residue: | 382 |
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| Sequence: | MNSTLFSRVENYSVHYNVSENSPFLAFENDDCHLPLAVIFTLALAYGAVIILGVSGNLAL
IIIILKQKEMRNVTNILIVNLSFSDLLVAVMCLPFTFVYTLMDHWVFGETMCKLNPFVQC
VSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYIGITVIWVLAVASSLPFVIYQILTD
EPFQNVSLAAFKDKYVCFDKFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRR
NNMMDKIRDSKYRSSETKRINVMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLL
FLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSK
TSLKQASPVAFKKISMNDNEKI
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| BDBM50065468 |
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| n/a |
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| Name | BDBM50065468 |
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| Synonyms: | 2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-1-yl-propoxy)-1-(3-piperidin-3-yl-propyl)-1H-benzoimidazole | CHEMBL61532 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H41ClN4O2 |
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| Mol. Mass. | 525.125 |
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| SMILES | Clc1ccc(OCc2nc3c(OCCCN4CCCCC4)cccc3n2CCCC2CCCNC2)cc1 |
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| Structure | 
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