| Reaction Details |
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 | Report a problem with these data |
| Target | Casein kinase I isoform gamma-2 |
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| Ligand | BDBM50519662 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1877798 (CHEMBL4379192) |
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| IC50 | >10000±n/a nM |
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| Citation |  Zhao, L; Li, Y; Wang, Y; Qiao, Z; Miao, Z; Yang, J; Huang, L; Tian, C; Li, L; Chen, D; Yang, S Discovery of 4 J Med Chem62:10691-10710 (2019) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Casein kinase I isoform gamma-2 |
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| Name: | Casein kinase I isoform gamma-2 |
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| Synonyms: | CK1G2 | CSNK1G2 | Casein kinase I | Casein kinase I gamma 2 | KC1G2_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47475.36 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_774313 |
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| Residue: | 415 |
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| Sequence: | MDFDKKGGKGETEEGRRMSKAGGGRSSHGIRSSGTSSGVLMVGPNFRVGKKIGCGNFGEL
RLGKNLYTNEYVAIKLEPIKSRAPQLHLEYRFYKQLSATEGVPQVYYFGPCGKYNAMVLE
LLGPSLEDLFDLCDRTFTLKTVLMIAIQLITRMEYVHTKSLIYRDVKPENFLVGRPGTKR
QHAIHIIDFGLAKEYIDPETKKHIPYREHKSLTGTARYMSINTHLGKEQSRRDDLEALGH
MFMYFLRGSLPWQGLKADTLKERYQKIGDTKRATPIEVLCENFPEEMATYLRYVRRLDFF
EKPDYDYLRKLFTDLFDRSGFVFDYEYDWAGKPLPTPIGTVHTDLPSQPQLRDKTQPHSK
NQALNSTNGELNADDPTAGHSNAPITAPAEVEVADETKCCCFFKRRKRKSLQRHK
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| BDBM50519662 |
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| n/a |
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| Name | BDBM50519662 |
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| Synonyms: | CHEMBL4438748 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H23N3O5 |
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| Mol. Mass. | 457.4779 |
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| SMILES | CN(C)c1ccc(cc1)C(=O)Nc1cccc(NC(=O)COc2ccc3c(c2)occc3=O)c1 |
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| Structure | 
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