| Reaction Details |
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 | Report a problem with these data |
| Target | D(3) dopamine receptor |
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| Ligand | BDBM50075359 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_58773 |
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| Ki | 50±n/a nM |
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| Citation |  Curtis, NR; Kulagowski, JJ; Leeson, PD; Ridgill, MP; Emms, F; Freedman, SB; Patel, S; Patel, S Synthesis and sar of 2- and 3-substituted 7-azaindoles as potential dopamine D4 ligands. Bioorg Med Chem Lett9:585-8 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| D(3) dopamine receptor |
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| Name: | D(3) dopamine receptor |
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| Synonyms: | DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3 |
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| Type: | n/a |
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| Mol. Mass.: | 44243.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 400 |
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| Sequence: | MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERAL
QTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILN
LCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTV
CSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQ
QTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRK
LSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHV
SPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
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| BDBM50075359 |
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| n/a |
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| Name | BDBM50075359 |
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| Synonyms: | 2-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrrolo[2,3-b]pyridine | CHEMBL347155 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H21ClN4 |
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| Mol. Mass. | 340.85 |
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| SMILES | Clc1ccc(cc1)N1CCN(CCc2cc3cccnc3[nH]2)CC1 |
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| Structure | 
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