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TargetTranscriptional activator protein LasR
LigandBDBM50351511
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1901853 (CHEMBL4404075)
EC50>200000±n/a nM
Citation Chbib, C Impact of the structure-activity relationship of AHL analogues on quorum sensing in Gram-negative bacteria. Bioorg Med Chem28:0 (2020) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Transcriptional activator protein LasR
Name:Transcriptional activator protein LasR
Synonyms:LASR_PSEAE | lasR
Type:PROTEIN
Mol. Mass.:26618.24
Organism:Pseudomonas aeruginosa
Description:ChEMBL_1475312
Residue:239
Sequence:
MALVDGFLELERSSGKLEWSAILQKMASDLGFSKILFGLLPKDSQDYENAFIVGNYPAAW
REHYDRAGYARVDPTVSHCTQSVLPIFWEPSIYQTRKQHEFFEEASAAGLVYGLTMPLHG
ARGELGALSLSVEAENRAEANRFMESVLPTLWMLKDYALQSGAGLAFEHPVSKPVVLTSR
EKEVLQWCAIGKTSWEISVICNCSEANVNFHMGNIRRKFGVTSRRVAAIMAVNLGLITL
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BDBM50351511
n/a
NameBDBM50351511
Synonyms:CHEMBL463321
TypeSmall organic molecule
Emp. Form.C12H19NO4
Mol. Mass.241.2836
SMILESCCCCCC(=O)CC(=O)N[C@H]1CCOC1=O |r|
Structure
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