| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50380892 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1935004 (CHEMBL4480763) |
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| Ki | 36±n/a nM |
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| Citation |  Leleu-Chavain, N; Baudelet, D; Heloire, VM; Rocha, DE; Renault, N; Barczyk, A; Djouina, M; Body-Malapel, M; Carato, P; Millet, R Benzo[d]thiazol-2(3H)-ones as new potent selective CB Eur J Med Chem165:347-362 (2019) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50380892 |
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| n/a |
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| Name | BDBM50380892 |
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| Synonyms: | CHEMBL2019090 | S-777469 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H27FN2O4 |
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| Mol. Mass. | 414.4699 |
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| SMILES | CCc1c(C)cc(C(=O)NC2(CCCCC2)C(O)=O)c(=O)n1Cc1ccc(F)cc1 |
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| Structure | 
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