| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 2 |
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| Ligand | BDBM50148351 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1977565 (CHEMBL4610700) |
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| EC50 | 1089±n/a nM |
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| Citation |  González-Gil, I; Zian, D; Vázquez-Villa, H; Hernández-Torres, G; Martínez, RF; Khiar-Fernández, N; Rivera, R; Kihara, Y; Devesa, I; Mathivanan, S; Del Valle, CR; Zambrana-Infantes, E; Puigdomenech, M; Cincilla, G; Sanchez-Martinez, M; Rodríguez de Fonseca, F; Ferrer-Montiel, AV; Chun, J; López-Vales, R; López-Rodríguez, ML; Ortega-Gutiérrez, S A Novel Agonist of the Type 1 Lysophosphatidic Acid Receptor (LPA J Med Chem63:2372-2390 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 2 |
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| Name: | Lysophosphatidic acid receptor 2 |
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| Synonyms: | EDG4 | LPA receptor 2 | LPA-2 | LPA2 | LPAR2 | LPAR2_HUMAN | Lysophosphatidic acid receptor 2 | Lysophosphatidic acid receptor Edg-4 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 39103.44 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1451385 |
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| Residue: | 351 |
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| Sequence: | MVIMGQCYYNETIGFFYNNSGKELSSHWRPKDVVVVALGLTVSVLVLLTNLLVIAAIASN
RRFHQPIYYLLGNLAAADLFAGVAYLFLMFHTGPRTARLSLEGWFLRQGLLDTSLTASVA
TLLAIAVERHRSVMAVQLHSRLPRGRVVMLIVGVWVAALGLGLLPAHSWHCLCALDRCSR
MAPLLSRSYLAVWALSSLLVFLLMVAVYTRIFFYVRRRVQRMAEHVSCHPRYRETTLSLV
KTVVIILGAFVVCWTPGQVVLLLDGLGCESCNVLAVEKYFLLLAEANSLVNAAVYSCRDA
EMRRTFRRLLCCACLRQSTRESVHYTSSAQGGASTRIMLPENGHPLMDSTL
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| BDBM50148351 |
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| n/a |
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| Name | BDBM50148351 |
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| Synonyms: | CHEMBL117529 | [3-((Z)-Octadec-9-enoylamino)-propionyl]-phosphonic acid |
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| Type | Small organic molecule |
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| Emp. Form. | C21H40NO5P |
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| Mol. Mass. | 417.5198 |
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| SMILES | CCCCCCCC\C=C/CCCCCCCC(=O)NCCC(=O)P(O)(O)=O |
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| Structure | 
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